BDBM264085 2-[3-[2-(4-chlorophenyl)propan- 2-yl]-5-hydroxypyrazol-1- yl]pyridine-4-carboxylic acid::US10173996, Example 170::US9604961, Example 170::US9714230, 170::US9908865, Example 170

SMILES CC(C)(c1cc(O)n(n1)-c1cc(ccn1)C(O)=O)c1ccc(Cl)cc1

InChI Key InChIKey=KZVFIAJADGKVPK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 264085   

TargetLysine-specific demethylase 2B(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 264085BDBM264085(2-[3-[2-(4-chlorophenyl)propan- 2-yl]-5-hydroxypyr...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 264085BDBM264085(2-[3-[2-(4-chlorophenyl)propan- 2-yl]-5-hydroxypyr...)
Affinity DataIC50: 5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
US Patent