BDBM2711 3-(1,2,3,4-Tetrahydropyrazino[1,2-a]indol-10-yl)-4-(1-methyl-3-indolyl)-1H-pyrrole-2,5-dione::3-(1-methyl-1H-indol-3-yl)-4-{1H,2H,3H,4H-pyrazino[1,2-a]indol-10-yl}-2,5-dihydro-1H-pyrrole-2,5-dione::Bisindolylmaleimide deriv. 17::ROCHE screening, 63
SMILES Cn1cc(C2=C(C(=O)NC2=O)c2c3CNCCn3c3ccccc23)c2ccccc12
InChI Key InChIKey=WGLDKILPHLGLGQ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 2711
Affinity DataIC50: 540nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:IC50 determinations for TBK1 were performed with the KinEASE-STK assay from Cisbio according to the manufacturer's instructions. A biotinylated s...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair