BDBM27251 indan derivative, 1::tert-butyl 2-(2-benzenesulfonamido-2,3-dihydro-1H-inden-5-yl)-1H-indole-1-carboxylate

SMILES CC(C)(C)OC(=O)n1c(cc2ccccc12)-c1ccc2CC(Cc2c1)NS(=O)(=O)c1ccccc1

InChI Key InChIKey=ODJWHQQYADUVIQ-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 27251   

TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(indan derivative, 1 | tert-butyl 2-(2-benzenesulfo...)
Affinity DataEC50:  190nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(indan derivative, 1 | tert-butyl 2-(2-benzenesulfo...)
Affinity DataEC50:  210nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(indan derivative, 1 | tert-butyl 2-(2-benzenesulfo...)
Affinity DataEC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed