BDBM272827 (S)-2-((1- ([1,2,4]triazolo[1,5- a]pyridin-7-yl)-8,9- dihydro-7H-6-oxa- 2,9a- diazabenzo[cd]azulen- 4-yl)amino)-2- cyclopropylacetamide::US10065970, Compound 132::US10435414, Compound 132

SMILES NC(=O)[C@@H](Nc1cc2OCCCn3c(nc(c1)c23)-c1ccn2ncnc2c1)C1CC1

InChI Key InChIKey=XLIDNDQXWYBDHM-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 272827   

LigandPNGBDBM272827((S)-2-((1- ([1,2,4]triazolo[1,5- a]pyridin-7-yl)-8...)
Affinity DataKi:  1.60nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

LigandPNGBDBM272827((S)-2-((1- ([1,2,4]triazolo[1,5- a]pyridin-7-yl)-8...)
Affinity DataKi:  1.60nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent