BDBM277159 US10072003, Example 7-1::US10072003, Example 7-2

SMILES CC(N1CCc2c(C1)nc(cc2-c1ccc(F)cc1F)C(N)=O)c1cnnn1C

InChI Key InChIKey=RGCDODFOMCDOAW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 277159   

TargetMetabotropic glutamate receptor 2(Human)
TBA

US Patent
LigandPNGBDBM277159(US10072003, Example 7-2 | US10072003, Example 7-1)
Affinity DataIC50: 3.74E+4nMAssay Description:The utility of the compounds of the invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR2 activity, may be demon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 2(Human)
TBA

US Patent
LigandPNGBDBM277159(US10072003, Example 7-2 | US10072003, Example 7-1)
Affinity DataIC50: 4.59E+4nMAssay Description:The utility of the compounds of the invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR2 activity, may be demon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent