BDBM284998 N-[2,4-difluoro-5-[2-methyl-6-(1- methylpyrazol-4-yl)-1-oxoisoquinolin-4-yl] phenyl]methanesulfonamide::US10023592, Example 43
SMILES Cn1cc(cn1)-c1ccc2c(c1)c(cn(C)c2=O)-c1cc(NS(C)(=O)=O)c(F)cc1F
InChI Key InChIKey=GPNYKSPNXFZEEW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 284998
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair