BDBM30285 indole-based 6-membered lactam, (S)-4a

SMILES NC[C@H]1Cn2c(cc3ccc(cc23)C(=O)Nc2cccnc2)C(=O)N1

InChI Key InChIKey=MMWVUKRVNHSCOU-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 30285   

TargetMAP kinase-activated protein kinase 2 [41-364](Human)
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM30285(indole-based 6-membered lactam, (S)-4a)
Affinity DataIC50: 2.30E+3nMpH: 7.6 T: 2°CAssay Description:Diluted compounds and activated GST-MK2 were incubated in neutravidin coated plates (Pierce) in reaction buffer containing biotinylated GST-LSP1 and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2009
Entry Details Article
PubMed