BDBM319074 US10173991, Example 117::methyl N-{3-[2- ({[(cyclopropyl- carbamoyl)methyl] carbamoyl} (methanesulfonyl) methyl)-5-fluoro- 1,3-benzothiazol- 6-yl]phenyl} carbamate

SMILES COC(=O)Nc1cccc(c1)-c1cc2sc(nc2cc1F)C(C(=O)NCC(=O)NC1CC1)S(C)(=O)=O

InChI Key InChIKey=WBPIDSFDCHYSFP-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 319074   

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM319074(US10173991, Example 117 | methyl N-{3-[2- ({[(cycl...)
Affinity DataIC50: 4nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
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Date in BDB:
5/15/2019
Entry Details
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