BDBM328660 (S)-2,2,2-trichloroethyl (2- (cyclopropanecarboxamidomethyl)- 4-((4-fluorophenyl)sulfonyl)-3,4- dihydro-2H-benzo[b][1,4]oxazin-6- yl)carbamate::US9663502, 30T
SMILES Fc1ccc(cc1)S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OCC(Cl)(Cl)Cl)cc12
InChI Key InChIKey=HPATWWMACUQYLQ-INIZCTEOSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 328660
Affinity DataIC50: 8.09nMAssay Description:The compounds of the invention inhibit RORgammaT activity. Activation of RORgammaT activity can be measured using, e.g., a biochemical TR-FRET assay....More data for this Ligand-Target Pair