BDBM345654 Ethanesulfonic acid [2-(2-methoxy- phenyl)-6-(1-methyl-6-oxo-1,6- dihydro-pyridin-3-yl)-pyrimidin-4- yl]-amide::US10202360, Example 199

SMILES CCS(=O)(=O)Nc1cc(nc(n1)-c1ccccc1OC)-c1ccc(=O)n(C)c1

InChI Key InChIKey=JOUUJLPBRZMOCX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 345654   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM345654(US10202360, Example 199 | Ethanesulfonic acid [2-(...)
Affinity DataIC50: 2.75E+3nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent