BDBM347135 2-(4-((cyclopropylmethyl)(3-(4-methyl piperazin-1-yl)phenyl)amino)phenoxy) pyrido[3,4-d]pyrimidin-4-ol::US10202381, Example 142::US10208039, Example 142

SMILES CN1CCN(CC1)c1cccc(c1)N(CC1CC1)c1ccc(Oc2nc(O)c3ccncc3n2)cc1

InChI Key InChIKey=KEECQYWHLQJXND-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 347135   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM347135(2-(4-((cyclopropylmethyl)(3-(4-methyl piperazin-1-...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent