BDBM369498 Intermediate 79: tert-butyl ((1R, 2S)-2-phenylcyclopropyl)(piperidin-4-yl)carbamate::US10233152, Example 36

SMILES FC(F)(F)C(=O)N1CCC(CC1)N[C@@H]1C[C@H]1c1ccccc1

InChI Key InChIKey=DGWVIICLBIXNBC-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369498   

TargetLysine-specific histone demethylase 1A(Human)
Mirati Therapeutics

US Patent
LigandPNGBDBM369498(Intermediate 79: tert-butyl ((1R, 2S)-2-phenylcycl...)
Affinity DataIC50: 33nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
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Date in BDB:
12/27/2019
Entry Details
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