BDBM383590 (1-(cyclopropylmethyl)piperidin-3-yl)(3-methoxyphenyl)methanone::US10280149, Example 109a

SMILES COc1cccc(c1)C(=O)[C@@H]1CCCN(CC2CC2)C1

InChI Key InChIKey=VNWQPWKGTWDASM-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383590   

TargetLysine-specific demethylase 2B(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 383590BDBM383590((1-(cyclopropylmethyl)piperidin-3-yl)(3-methoxyphe...)
Affinity DataIC50: 1.41E+4nMAssay Description:Full length KDM2B was cloned, expressed, and purified to homogeneity. Compound inhibition of KDM2B demethylase activity was assessed by monitoring th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
US Patent