BDBM385792 US10287286, Example 195::cyclopropylmethyl N-[5-(4- cyano-3-fluorophenyl)- [1,2,4]triazolo[1,5-a]pyridin- 7-yl]carbamate

SMILES Fc1cc(ccc1C#N)-c1cc(NC(=O)OCC2CC2)cc2ncnn12

InChI Key InChIKey=HALMVMOOYFNWCX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 385792   

TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM385792(US10287286, Example 195 | cyclopropylmethyl N-[5-(...)
Affinity DataIC50:  14nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent