BDBM437465 2-Benzyl-4-(1,5-dimethyl-6-oxo-1,6-dihydro-pyridin-3- yl)-2H-pyrazole-3-carboxylic acid ethyl ester::US10617680, Example 199::US11020380, Example 199

SMILES CCOC(=O)c1c(cnn1Cc1ccccc1)-c1cc(C)c(=O)n(C)c1

InChI Key InChIKey=OVKVQAVEOBZLKZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437465   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437465(2-Benzyl-4-(1,5-dimethyl-6-oxo-1,6-dihydro-pyridin...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437465(2-Benzyl-4-(1,5-dimethyl-6-oxo-1,6-dihydro-pyridin...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent