BDBM437569 Ethanesulfonic acid 2-[4-(4-cyclopropyl-1-methyl-6-oxo- 1,6-dihydro-pyridin-3-yl)-pyrazol-1-yl]-benzoylamide::US10617680, Example 303::US11020380, Example 303

SMILES CCS(=O)(=O)NC(=O)c1ccccc1-n1cc(cn1)-c1cn(C)c(=O)cc1C1CC1

InChI Key InChIKey=BJQOLJWCFFVSBX-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437569   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 437569BDBM437569(Ethanesulfonic acid 2-[4-(4-cyclopropyl-1-methyl-6...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2021
Entry Details
US Patent

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 437569BDBM437569(Ethanesulfonic acid 2-[4-(4-cyclopropyl-1-methyl-6...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent