BDBM446939 3-[6-(3- thienyl)imidazo [1,2-a]pyrazin- 3-yl]phenol::US10688093, Compound 388_0284_0074::US11701353, Compound 388_0284_0074

SMILES Oc1cccc(c1)-c1cnc2cnc(cn12)-c1ccsc1

InChI Key InChIKey=UBQAKVDLEIHDNI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 446939   

TargetTyrosine-protein kinase Fyn(Human)
Pathways Neuro Pharma

US Patent
LigandPNGBDBM446939(3-[6-(3- thienyl)imidazo [1,2-a]pyrazin- 3-yl]phen...)
Affinity DataIC50: 2.52E+3nMAssay Description:The assay procedure determines the IC50 of each potential FYN kinase inhibitor by measuring the enzyme catalyzed ATP-dependent phosphorylation of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details
US Patent