BDBM473526 US10844044, Example 266::US10844044, Example 362

SMILES Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1

InChI Key InChIKey=RWDXQFHWSULJBR-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 473526   

TargetWD repeat-containing protein 5(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 473526BDBM473526(US10844044, Example 362 | US10844044, Example 266)
Affinity DataKi:  0.720nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2021
Entry Details
US Patent

TargetWD repeat-containing protein 5(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 473526BDBM473526(US10844044, Example 362 | US10844044, Example 266)
Affinity DataKi:  16nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2021
Entry Details
US Patent