BDBM50005364 (3S,4R)3-Methyl-3-(3-methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bicyclo[2.2.1]heptane::CHEMBL171721
SMILES Cc1noc(n1)C1(C)CN2CCC1C2
InChI Key InChIKey=KCRQRKFNDXRLPR-UHFFFAOYSA-N
Data 3 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50005364
TargetMuscarinic acetylcholine receptor M1(RAT)
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Compound was tested in vitro for depolarizing response on the rat superior cervical ganglion(mediated by muscarinic acetylcholine receptor M1)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:In vitro negative chronotropic effect of the compound on electrically driven guinea pig atria(mediated by muscarinic acetylcholine receptor M2)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Compound was tested in vitro for the contraction of guinea pig myenteric plexus preparation (mediated by muscarinic acetylcholine receptor M3)More data for this Ligand-Target Pair