BDBM50006842 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-3-(3-isopropoxy-phenyl)-3H-quinazolin-4-one::CHEMBL37312
SMILES CC(C)Oc1cccc(c1)-n1c(CCc2c[nH]c3ccc(Br)cc23)nc2ccccc2c1=O
InChI Key InChIKey=KUECXUACQOYKNB-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50006842
Affinity DataIC50: 9.30nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]-labeled gastrin binding to gastrin/cholecystokinin type B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Antagonistic activity against cholecystokinin type B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibition of [125I]-CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair