BDBM50055267 CHEMBL3323682
SMILES CCCCCCC(C)(C)c1cc(O)cc(OCCCCCCCC(=O)NCC=C)c1
InChI Key InChIKey=IDSPJWVYIKNBSP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50055267
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataIC50: 2.39E+4nMAssay Description:Antagonist activity against human recombinant TRPV1 expressed in HEK293 cells assessed as reduction in capsaicin-induced intracellular calcium respon...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Antagonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as reduction in isothiocynate-induced increase in intracellular calci...More data for this Ligand-Target Pair
Affinity DataEC50: 138nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 6.90E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluorescence assayMore data for this Ligand-Target Pair