BDBM50094505 2-((4-phenylpiperazin-1-yl)methyl)-1H-indole-5-carbonitrile::2-(4-Phenyl-piperazin-1-ylmethyl)-1H-indole-5-carbonitrile::CHEMBL140099
SMILES N#Cc1ccc2[nH]c(CN3CCN(CC3)c3ccccc3)cc2c1
InChI Key InChIKey=TWVIJESEEXGVPP-UHFFFAOYSA-N
Data 13 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 50094505
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4.4 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2S expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Laboratoire De Chimie Th�Rapeutique
Curated by ChEMBL
Laboratoire De Chimie Th�Rapeutique
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D3 in CHO cell membraneMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Laboratoire De Chimie Th�Rapeutique
Curated by ChEMBL
Laboratoire De Chimie Th�Rapeutique
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to human D3R assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2L expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Binding affinity to human D2R assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Displacement of [3H]SCH 23990 from dopamine receptor D1 in porcine striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Displacement of [3H]SCH-23390 from Dopamine receptor D1 of bovine striatal membranesMore data for this Ligand-Target Pair