BDBM50126548 4-{4-[Benzenesulfonyl-(3H-imidazol-4-ylmethyl)-amino]-phenyl}-piperazine-1-carbothioic acid phenethyl-amide::CHEMBL286899

SMILES O=S(=O)(N(Cc1cnc[nH]1)c1ccc(cc1)N1CCN(CC1)C(=S)NCCc1ccccc1)c1ccccc1

InChI Key InChIKey=ZYNGWCIWJAOSGO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50126548   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bovine)
Centre De Recherche Pierre Fabre

Curated by ChEMBL

LigandBDBM50126548(4-{4-[Benzenesulfonyl-(3H-imidazol-4-ylmethyl)-ami...)Copy SMILESCopy InChI

Affinity DataIC50: 100nMAssay Description:Inhibit of purified bovine Farnesyl protein transferase.More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/9/2012
Entry Details Article
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