BDBM50152059 3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-ethyl-pentyl)-1-methyl-1,2,3,7-tetrahydro-purin-6-one::CHEMBL363023

SMILES CCCCC(CC)n1c(CC)nc2N(CN(C)C(=O)c12)c1ccc(Cl)cc1Cl

InChI Key InChIKey=YDPLDDJWUQCPNL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50152059   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152059(3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-ethyl-pentyl)...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed