BDBM50153533 3-(2,6-Dichloro-phenyl)-5-[2-(2-methoxy-phenyl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide::CHEMBL365721
SMILES CCN(CC)c1ccc(NC(=O)c2c(CCc3ccccc3OC)onc2-c2c(Cl)cccc2Cl)cc1
InChI Key InChIKey=RBBWIQSVRIEEHC-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50153533
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 389nMAssay Description:Ability to displace [125I]-ghrelin from cloned human GHS-R expressed in CHO-K cells was determined (Kd of ghrelin is 0.4 nM)More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 714nMAssay Description:Ability to inhibit ghrelin induced increase in intracellular [Ca2+] in CHO-K cells was determined by FLIPR assayMore data for this Ligand-Target Pair