BDBM501890 US11028075, Example 23
SMILES Fc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1
InChI Key InChIKey=BAZPFEMDCRMFGC-OEOAZWSVSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 501890
Affinity DataIC50: 1.63nMAssay Description:The following voltage clamp electrophysiology studies are performed on representative compounds using cells heterologously expressing Nav1.7 or Nav1....More data for this Ligand-Target Pair
Affinity DataIC50: 1.21nMAssay Description:Saturation experiments. A competitive NaV1.7 inhibitor having a methyl group is tritiated. Three tritiums are incorporated in place of methyl hydroge...More data for this Ligand-Target Pair