BDBM50238037 CHEMBL4082235

SMILES CN(CCCNc1cc(=O)oc2ccccc12)C(=O)c1cccs1

InChI Key InChIKey=GHTHAUJPTBYQOJ-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50238037   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50238037(CHEMBL4082235)
Affinity DataIC50:  810nMAssay Description:Inhibition of human BRD4-BD1 (49 to 170 residues) expressed in Escherichia coli BL21(DE3) using N-C:SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHRKVGG-K...More data for this Ligand-Target Pair