Affinity DataKi: 0.0180nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:In vitro inhibition of [3H]NT binding to porcine striatal Neurotensin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]-Tyr(3)-NT to human Neurotensin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 3More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.160nMAssay Description:In vitro inhibition of [3H]-NT binding to human striatal Neurotensin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 0.0100nMAssay Description:Agonist activity at rat NTS1 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as inhibition of SR142948a-induced calcium release by FLIPR assayMore data for this Ligand-Target Pair