BDBM50324797 3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-yl)propanamide::3-[1-(4-Chloro-benzyl)-1H-indol-3-yl]-N-pyridin-4-yl-propionamide::CHEMBL185140::N-(pyridin-4-yl)-3-[1-(4-chlorobenzyl)indol-3-yl]-propanamide

SMILES Clc1ccc(Cn2cc(CCC(=O)Nc3ccncc3)c3ccccc23)cc1

InChI Key InChIKey=KTMXBAQZQLHSIQ-UHFFFAOYSA-N

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50324797   

TargetVascular endothelial growth factor receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant KDR after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant YES after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of recombinant JAK3 after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant c-Abl after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant aurora A after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Pim1 after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant HIPK1 after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant TrkA after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50324797(3-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N-(pyridin-4-...)
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of recombinant JAK2 after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed