BDBM50327538 3-((4-bromophenethylamino)methyl)-2-(thiophen-3-yl)quinolin-7-ol::CHEMBL1257491
SMILES Oc1ccc2cc(CNCCc3ccc(Br)cc3)c(nc2c1)-c1ccsc1
InChI Key InChIKey=AOKMPEUHFZVJJB-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50327538
Affinity DataIC50: 280nMAssay Description:Agonist activity at mouse TGR5 receptor expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair