BDBM50334752 3-(Phenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl::CHEMBL1642880

SMILES O=S(=O)(c1n[nH]c2ccc(NC3CCNCC3)cc12)c1ccccc1

InChI Key InChIKey=YLOKQWYOYZLCMX-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50334752   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334752(3-(Phenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-LSD from cloned human 5-HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334752(3-(Phenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5...)
Affinity DataIC50:  125nMAssay Description:Antagonist activity at cloned human 5-HT6 receptor expressed in human HeLa cells assessed as inhibition of 5HT-induced cyclic AMP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed