BDBM50347738 CHEMBL1803076

SMILES CCCNC1=NC(=Cc2ccccc2O)C(=O)N1C

InChI Key InChIKey=IHKPHJVJQJQFDE-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50347738   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347738BDBM50347738(CHEMBL1803076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged DYRK2 using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347738BDBM50347738(CHEMBL1803076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347738BDBM50347738(CHEMBL1803076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Mouse)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347738BDBM50347738(CHEMBL1803076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK3 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347738BDBM50347738(CHEMBL1803076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant Pim1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed