BDBM50412245 CHEMBL495095
SMILES CC(Oc1ccccc1CC=C)C1=NCCN1
InChI Key InChIKey=MNMDMCKHXVHLAW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50412245
Affinity DataKi: 28nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic Alpha-2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of human ERG expressed in HEK293 cells after 240 secs by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair