BDBM50416075 CHEMBL1086260
SMILES CC(C)N(c1ccccc1)S(=O)(=O)c1ccc(-c2ccc3n(ncc3c2)-c2ccc(F)cc2)c(c1)C(F)(F)F
InChI Key InChIKey=STMSGZQNLAWSTI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50416075
Affinity DataIC50: 15.8nMAssay Description:Displacement of fluorescent-labeled Dexamethasone from GR by fluorescent polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to ARMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Activity at GR in human A549 cells by NF-kappaB transrepression assayMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GR in human A549 cells transfected with luciferase gene linked to MMTV promoter assessed as luciferase transactivation activity a...More data for this Ligand-Target Pair
Affinity DataIC50: >2.51E+3nMAssay Description:Binding affinity to PRMore data for this Ligand-Target Pair