BDBM50509369 CHEMBL4548361

SMILES COc1cc(Br)cc2[nH]c(I)c(-c3cnc(-c4ccc[nH]4)o3)c12

InChI Key InChIKey=NDWPRZFOCQREKV-UHFFFAOYSA-N

Data  13 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 13 hits for monomerid = 50509369   

TargetMitogen-activated protein kinase 15(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase SIK3(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509369BDBM50509369(CHEMBL4548361)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed