BDBM50544595 CHEMBL4639199
SMILES FC(F)(F)c1ccc(Oc2ccc(CCNC(=O)C(=O)CCCc3ccccc3)cc2)nc1
InChI Key InChIKey=DZHZISUSQMPBJQ-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50544595
TargetPhospholipase A and acyltransferase 2(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT2 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 4(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT4 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair