BDBM508654 (R or S)-8-[2-(3,3-difluoroazetidin- 1-yl)propyl]-2,2-difluoro[1,3] dioxolo[4,5-h][1,2,4]triazolo[1,5-c] quinazolin-5-amine (faster eluting b)::US11046714, Example 93::US11046714, Example 94
SMILES CC(Cc1nc2c3ccc4OC(F)(F)Oc4c3nc(N)n2n1)N1CC(F)(F)C1
InChI Key InChIKey=ILIXALIZILTPHR-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 508654
Affinity DataKi: 4.10nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair