BDBM508710 (R or S)-8-[1-(3,5-difluorophenyl) piperidin-3-yl]-2,2-difluoro[1,3] dioxolo[4,5-h][1,2,4]triazolo[1,5- c]quinazolin-5-amine (faster eluting a)::US11046714, Example 144::US11046714, Example 145
SMILES Nc1nc2c3OC(F)(F)Oc3ccc2c2nc(nn12)C1CCCN(C1)c1cc(F)cc(F)c1
InChI Key InChIKey=HCVZIZVSGQBNBV-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 508710
Affinity DataKi: 1.20nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair