BDBM530338 WO2022064009, Compound 125

SMILES C[C@@H]1Cc2cnc(Nc3cnn(C)c3)nc2CN1C(=O)[C@@H]1CCN(C)C[C@H]1c1cccc(C)c1

InChI Key InChIKey=FLAUIOGBWZNNGG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 530338   

TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Human)
Janssen Pharmaceutica

WIPO

LigandBDBM530338(WO2022064009, Compound 125)Copy SMILESCopy InChI

Affinity DataIC50: 339nMAssay Description:Inhibition potencies of compounds were studied using an absorbance kinetic assay as described below. Compounds with potencies approaching the limit o...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/2/2022
Entry Details
Copy BDB DOIWIPO WO2022064009

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