BDBM530385 WO2022064009, Compound 162

SMILES CC(C)N1CC[C@@H]([C@H](C1)c1ccc(Cl)c(F)c1)C(=O)N1Cc2nc(NC3CCOCC3)ncc2C[C@H]1C

InChI Key InChIKey=KLPTVWQIHFFMLW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 530385   

TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Human)
Janssen Pharmaceutica

WIPO

LigandBDBM530385(WO2022064009, Compound 162)Copy SMILESCopy InChI

Affinity DataIC50: 112nMAssay Description:Inhibition potencies of compounds were studied using an absorbance kinetic assay as described below. Compounds with potencies approaching the limit o...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/2/2022
Entry Details
Copy BDB DOIWIPO WO2022064009

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