BDBM562148 Methyl 2-[[5-(methylcarbamoyl)-1-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)benzimidazol-2-yl]methyl]benzoate::US11401256, Example 41

SMILES CNC(=O)c1ccc2n(c(Cc3ccccc3C(=O)OC)nc2c1)-c1ccc2NC(=O)CCc2c1

InChI Key InChIKey=PYUHFNXNGPBDPL-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 562148   

TargetProtein cereblon(Human)
C4 Therapeutics

US Patent
LigandPNGBDBM562148(US11401256, Example 41 | Methyl 2-[[5-(methylcarba...)
Affinity DataKd:  68nMAssay Description:Process 1) Optimization of measurement parameters to minimize protein consumption and to minimize the dilution effect and the DMSO content 2) Titrati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
Go to US Patent