BDBM570673 US11897851, Compound 220

SMILES CCn1cncc1Cn2c(/C=C(C)/C(=O)O)cnc2CN5CCC(c4cccc(OCc3ccc(Cl)cn3)n4)CC5

InChI Key InChIKey=NKHNRXRCWQGQLJ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 570673   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM570673(US11897851, Compound 220)
Affinity DataEC50:  0.110nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
Go to US Patent