BDBM582139 US11518764, Compound I-148::US11518764, Compound I-149

SMILES CN(C1CCC(C1)c1cc(NC(=O)Cn2cc(-c3cc(Cl)c(O)c(c3)C(N)=O)c3c2ncn(C)c3=O)c(Cl)cn1)S(C)(=O)=O

InChI Key InChIKey=SMRXUPMPYRFVKV-UHFFFAOYSA-N

Data  2 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 582139   

TargetB-cell lymphoma 6 protein(Human)
Ontario Institute For Cancer Research (Oicr)

US Patent
LigandChemical structure of BindingDB Monomer ID 582139BDBM582139(US11518764, Compound I-149 | US11518764, Compound ...)
Affinity DataKd:  16.3nMAssay Description:SPR studies were performed using a Biacore™ T200 instrument (GE Health Sciences Inc.). The BCL6 BTB protein used in the FP assay was biotinylate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2023
Entry Details
US Patent

TargetB-cell lymphoma 6 protein(Human)
Ontario Institute For Cancer Research (Oicr)

US Patent
LigandChemical structure of BindingDB Monomer ID 582139BDBM582139(US11518764, Compound I-149 | US11518764, Compound ...)
Affinity DataKd:  20.9nMAssay Description:SPR studies were performed using a Biacore™ T200 instrument (GE Health Sciences Inc.). The BCL6 BTB protein used in the FP assay was biotinylate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2023
Entry Details
US Patent