BDBM602975 N-(4-(8-amino-3-isopropyl-5-(4-(methylamino)cyclohex-1-en-1-yl)imidazo[1,5-a]pyrazin-1-yl)-2,5-difluorophenyl)-1-(2-chlorophenyl)methanesulfonamide::US11649237, Example 196

SMILES CNC1CCC(=CC1)c1cnc(N)c2c(nc(C(C)C)n12)-c1cc(F)c(NS(=O)(=O)Cc2ccccc2Cl)cc1F

InChI Key InChIKey=OBJMHPJXWXAGSI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 602975   

LigandPNGBDBM602975(US11649237, Example 196 | N-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 9nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
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Date in BDB:
6/19/2023
Entry Details
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