BDBM614937 B4-2-1-2::US20230271937, Example B4-2-1-2

SMILES CC1(CNc2ncnc(N(Cc3ccc(cc3)C(F)(F)F)C3CC3)c2F)CCN(CC(N)=O)C[C@@H]1O

InChI Key InChIKey=GIKDUNNJLUOVMA-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 614937   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Nuevolution

US Patent
LigandPNGBDBM614937(US20230271937, Example B4-2-1-2 | B4-2-1-2)
Affinity DataEC50:  8.60nMAssay Description:The HEK293 cell line is co-transfected transiently with two plasmids, one with the RORγ ligand-binding domain fused to galactose-responsive tran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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