BDBM618593 US20230287003, Example 14a::US20230287003, Example 14b

SMILES C[C@@H]1CN(CCC1(F)F)c1ncc(Cl)c(Nc2ccc3n(C)c(=O)c4OCC[C@@H](Nc4c3c2)C2CC2)n1

InChI Key InChIKey=RVDRGDGQDMGINA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 618593   

TargetB-cell lymphoma 6 protein(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 618593BDBM618593(US20230287003, Example 14a | US20230287003, Exampl...)
Affinity DataIC50: 105nMAssay Description:Each 15 μL HTRF reaction in a 384-well black Proxiplate (Perkin Elmer) contained 1 nM Trx-6×His-BCL6 (in house-produced, human BCL6 BTB domain c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetB-cell lymphoma 6 protein(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 618593BDBM618593(US20230287003, Example 14a | US20230287003, Exampl...)
Affinity DataIC50: 182nMAssay Description:Each 15 μL HTRF reaction in a 384-well black Proxiplate (Perkin Elmer) contained 1 nM Trx-6×His-BCL6 (in house-produced, human BCL6 BTB domain c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent