BDBM623850 US11780845, Example 870::US11780845, Example 879

SMILES CC(=C)C(=O)Nc1ccc(cc1)-c1c(-c2ccc(cc2)C(=O)N2CCCC2)c2c(N)n[nH]c(=O)c2n1C

InChI Key InChIKey=INJACHHWMCOWPY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 623850   

TargetFibroblast growth factor receptor 2(Human)
Relay Therapeutics

US Patent
LigandPNGBDBM623850(US11780845, Example 879 | US11780845, Example 870)
Affinity DataIC50: 1.05E+4nMAssay Description:Compounds of the present invention were also tested in a FGFR2 Biochemical Caliper Assay. Compounds were prepared in 10 mM DMSO solution and serially...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 2(Human)
Relay Therapeutics

US Patent
LigandPNGBDBM623850(US11780845, Example 879 | US11780845, Example 870)
Affinity DataIC50: 1.05E+4nMAssay Description:Compounds of the present invention were also tested in a FGFR2 Biochemical Caliper Assay. Compounds were prepared in 10 mM DMSO solution and serially...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
Go to US Patent