BDBM683230 4-(5-(3-amino-8- azabicyclo[3.2.1] octane-8-yl)-8-(6- fluorobenzo[c] [1,2,5]oxadiazole- 5-yl)imidazolo [1,2-c]pyrimidin- 7-yl)-2- fluorobenzonitrile::US20240216357, Example 186

SMILES NC1CC2CCC(C1)N2c1nc(-c2ccc(C#N)c(F)c2)c(-c2cc3nonc3cc2F)c2nccn12

InChI Key InChIKey=NVYRYSSBYQTMOH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 683230   

TargetLysine-specific histone demethylase 1A(Human)
Sichuan Huiyu Pharmaceutical

US Patent
LigandPNGBDBM683230(US20240216357, Example 186 | 4-(5-(3-amino-8- azab...)
Affinity DataIC50: 17.3nMAssay Description:The effects of compounds on LSD1 enzyme activity are detected by an HTRF technology to evaluate their inhibition levels on LSD1 enzyme activity. Firs...More data for this Ligand-Target Pair
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Date in BDB:
10/11/2024
Entry Details
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