BDBM725692 WO2017214367, Example 64::US20250074910, Control compound 1

SMILES CC(C)c1ncncc1-c1cc(F)ccc1Oc1cncnc1N1CC2(CN(CC3CCC4(CC3)OCCO4)C2)C1

InChI Key InChIKey=PFXYDBYVJDWJFS-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 725692   

TargetHistone-lysine N-methyltransferase 2A(Human)
Hitgen

US Patent
LigandChemical structure of BindingDB Monomer ID 725692BDBM725692(WO2017214367, Example 64 | US20250074910, Control ...)
Affinity DataIC50: 156nMAssay Description:The inhibition of Menin/MLL-4-43 peptide interaction by small molecule inhibitors was quantitatively detected by fluorescence polarization competitio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/9/2025
Entry Details
US Patent