BDBM728917 US20250092064, Example 104

SMILES CCOC(=O)CC(c1cc(CN2C[C@@H](CC)Oc3cccnc3[C@@H]2C)c2ccn(C(=O)OC(C)(C)C)c2c1)c1cc(C2CC2)c2c(nnn2C)c1C

InChI Key InChIKey=RHTNMYBSHRZARS-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 728917   

LigandChemical structure of BindingDB Monomer ID 728917BDBM728917(US20250092064, Example 104)
Affinity DataIC50: 20nMAssay Description:The inhibitory activity of test compounds on the binding between Nrf2 and Keap1 was determined by fluorescence polarization. A solution of 50 mM Tris...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/25/2025
Entry Details
US Patent